China Arctiin Opanga ndi ogulitsa | Chenlv

Arctiin

Kufotokozera Kwachidule:

Arctiin ndi yogwira lignin zikuluzikulu zipatso za burdock chomera A. lappa. Zimasonyezanso amphamvu mavairasi oyambitsa ntchito ndi fuluwenza A HIV ndi zotsatira odana ndi yotupa ndi kucheperachepera yopanga okusayidi nitric ndi cytokines ovomereza-yotupa.


mankhwala Mwatsatanetsatane

Tags mankhwala

CAS No .:  20362-31-6

Latin dzina: Arctium lappa L.

Part ntchito:  zipatso

Maonekedwe:  chikasu bulauni chabwino ufa

Maselo chilinganizo:  C27H34O11

Maselo Kulemera kwake:  534,55

Mayeso njira:  HPLC

mfundo:

1.Arctiin10%

2.Arctiin20%

3.Arctiin40%

Arctigenin (AR) ndi glycoside ake, arctiin, ndizo awiri yogwira zosakaniza wa Arctium lappa L (A lappa), wotchuka mankhwala therere ndi thanzi enaake samasowa mu Asia. Mu zaka zapitazi, zigawo bioactive ku lappa A kuti chidwi ofufuza chifukwa zawo zotsatira zingamuthandize achire. M'nkhani pano, ife cholinga chake kupereka mwachidule za mankhwala a AR ndi arctiin, kuganizira zotsatira odana ndi yotupa zawo, katundu pharmacokinetics ndi efficacies matenda. Poyerekeza acrtiin, AR inanena kwambiri zimene bioactive chigawo cha A lappa mu ambiri a maphunziro. AR akusonyeza amphamvu ntchito odana ndi yotupa ndi inhibiting inducible nitric okusayidi synthase (iNOS) kudzera kusinthasintha mawu a cytokines angapo. Chifukwa zotsatira zake amphamvu odana ndi yotupa, AR ikhale angathe achire pawiri ndi onse pachimake kutupa ndi matenda osiyanasiyana aakulu. Komabe, maphunziro pharmacokinetic anasonyeza glucuronidation yaikulu ndi hydrolysis wa AR mu chiwindi, intestine ndi madzi a m'magazi, amene chingatilepheretse ake mu pompo-pompo ndi matenda efficacy pambuyo makonzedwe m'kamwa. Zochokera kuwunikira makhalidwe pharmacological ndi pharmacokinetic wa AR, pharmacokinetic patsogolo ndi maphunziro pharmacodynamic wa AR kudzera zodutsa njira makonzedwe ali akatswiri kulimbikitsa mphamvu yake kutumikira monga nthumwi achire komanso abwino bioactive chikhomo chifukwa lappa A.

Mankhwala wazolongedza:  25kg / ng'oma

Nthawi n'loonadi: zaka 2


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