14 Melemo ea Icariin

Icariin ke sebele ka holimo lethathamong leshome ba a tlatsana le hore ke nka ea ka. Ke ile ka reka mefuta e sa tsoaneng tse ngata tsa ena ho fumana ea molemo ka ho fetisisa.

Icariin ke eng?

Icariin ke tšobotsi e sebetsang flavonoid karolo ea Epimedium dimela mefuta tsejoang Horny Pōli Weed. Sefa tloha dimela tsena Ke khale ho sebelisoa ka setso Chinese Medicine bakeng sa ho matlafatsa libido le mosebetsi motona thobalano

Ka lebaka la kabo ea lona atile le mokhatlo oa 'meleng ho kopanyelletsa le boko, icariin lipontsuoa hole-ho tloha mesebetsi likokoana-hloko tse kang antioxidant le litla-ba khahlanong le a hlabang, neuroprotection, mosebetsi-ba khahlanong le hlahala, hammoho le ho khothalletsa bophelo bo botle ba ka kakaretso ka pelong, masapo,' me mefuta e fapaneng ya makala tse ling.

Experience Joe o Ka Horny Pōli Weed

Icariin ke o mong oa a tlatsana le ke e ratang ka 'me ke nka hore ho PDE5 inhibiting thepa. Ho tshepahala eketsa phallo ea mali ho pholletsa le 'mele' me o moholo bakeng sa ho eketsa mamello ho carbs.

Ho ntlafatsa tshebetso dikopanothutano le 'na le e leng khahlanong le a hlabang.

Melemo Bophelo ba Icariin

1.Improves Erectile ho se sebetse le eketsa Sex Drive
2. fokotsa Dementia le kgothaletsa dikopanothutano tsa Function
3. Icariin ke Neuroprotective le e Khothalletsa Neurogenesis
4. lowers Khatello ea Kelello le Melao e Antidepressant e
5. di hlohleletsago Bone Kgolo le Repair
6. e Khothalletsa Heart Bophelo
7. di hlohleletsago sebopeho Mali Sejana
8. hlahisa Anti-Kankere Liphello
9. Icariin ke Anti-a hlabang le Immunoprotective
10. Na Loantša Mokhathala
11. Sireletsa DNA le tieho ho Tsofala
12. Na Thusa maqoqomete a makhopho
13. Na Thusa pele ho nako mora ho ntsha peo
14. Na Fight Jetlag
1.Improves Erectile ho se sebetse le eketsa Sex Drive

Icariin thibela phosphodiesterase mofuta 5 (PDE5), e potlakisang tsebetso ea lik'hemik'hale hore roba fatše cyclic guanosine monophosphate (cGMP).

PDE5 thibelo di hlohleletsago le NO / cGMP tseleng le ho ntlafatsa mosebetsi ikatisa ka dikai liphoofolo.

Sena ke ka ntlha ya go eketseha cGMP le oxide e nitric maemo eo lebisa boreleli mesifa boikhathollo, o pharalla ea methapo ea mali le tse eketsehileng phallo ea mali ho botoneng ba, bebofatswe tsogelwa.

kalafo foleng la icariin ile a bontšoa ho thibela penile boreleli lefu mesifa seleng ea ka lithuto tsa multiple liphoofolo.

Ho phaella moo, icariin ile bontšoa haholo eketsa pelvic methapo ea kutlo bolelele ha rutehileng le likhechana methapo ea kutlo, e leng se bontšang hore ho ka 'na ntlafatsa penile tsosoloso ka batho.

Icariin ne a boetse a bontša ho eketsa mahala testosterone maemo ka likhoto.

Ho etsa lipatlisiso ho bontša hore maemo a phahameng a testosterone ba correlated le eketseha takatso ea ho kopanela liphate ka ho ba batona ba seng ba hōlile 'me tse tšehali, a fana ka maikutlo hore icariin e ka sebetsa jwalo ka e aphrodisiac tlhaho ka batho ba nang le libido qephe.

2. fokotsa Dementia le kgothaletsa dikopanothutano tsa Function

Icariin hlahisa mosebetsi-ba khahlanong le amyloid ka lithuto tse ngata tsa liphoofolo.

Beta-amyloid peptides (Aβ) ke liprotheine tse bakang pakellanang sebopeho le ho senya seleng ea ka lefu la Alzheimer.

Icariin ile bontšoa haholo fokotseha β-amyloid-hlohlelletsoa toxicity ka Rat adrenal lisele tse embryonic (by inhibiting ga tau protheine hyperphosphorylation, senotlolo sa likokoana-hloko lesupa ya lefu la Alzheimer).

Sena ke le monyetla ka lebaka la ho Tshebediso ya ya PI3K / Akt tseleng, tseo o phetha karolo ea bohlokoa ka ho pholoha seleng.

Icariin hape hlahisa liphello sireletsang khahlanong le haella ho ithuta le ho memori kapa ka dikai liphoofolo.

Icariin ntlafala dementia 'ka likhoto aluminium-tahiloe ka ho fokotsa tšenyo e oxidative le β-amyloid mobung ka hippocampus ena. Hona ke karolo e loketseng ho tse eketsehileng superoxide dismutase (SOD), e potlakisang tsebetso ea lik'hemik'hale hore ho fokotsa tšenyo e oxidative.

Ka dikai Rat le ho ruruha hlohlelletsoa boko, nako e khutsoanyane kalafo icariin ile a fumanoa a ho ntlafatsa tlhaloganya sebaka ho ithuta le ho memori kapa bokhoni. e le hantle ena e nahana hore ke ka lebaka la theola ya ea tse ling lan-hlabang (TNF-alpha, le IL-B hammoho le Cox-2, e potlakisang tsebetso ea lik'hemik'hale le boikarabelo ba ho feberu, ho ruruha, 'me bohloko).

Icariin ka boela hatella neuroinflammation ke inhibiting le Tshebediso ya ya microglia, lisele tse macrophage-joaloka ka boko ba tsamaiso ea methapo e phetha karolo ea bohlokoa ka ho qapa le neuroinflammatory karabo.

The-ba khahlanong le a hlabang phello ea icariin ka ngotsoe ke thibelo ea eona ea NF-κB le p38 MAPK litseleng, tse amehang microglia le proinflammatory lesupa Tshebediso ya.

ho ithuta e 'ngoe phoofolo ile a bontša hore icariin fokotseha fokotseha dikopanothutano ke eketseha BDNF le receptor tyrosine lona kinase TrkB.

BDNF ke le palokatiso neurotrophic amehang dirisa tlhaloganyo, synaptic plasticity, le ho pholoha neuronal.

Ka likhoto le setorouku, Icariin sireletsa khahlanong ditlhaelo dikopanothutano ke eketseha acetylcholine metabolism ka hippocampus, e leng neurotransmitter senotlolo amehang ho ithuta le ho hopola.

Ho phaella moo, Icariin ka khona ho ntlafatsa mosebetsi dikopanothutano dessyecik tlhotlheletso ya NO / cGMP tseleng. maemo e phahameng ea cGMP le oxide e nitric (ka tsela icariin thibelo ea PDE5) ntlafatsa boko phallo ea mali, synaptic plasticity, neurovascular ho se sebetse, 'me β-amyloid ntsha ho tswa hippocampus (setsi memoring ya) le cortex.

Ka lebaka lona matla-ba khahlanong le a hlabang, antioxidative le mosebetsi-ba khahlanong le amyloid bokong, icariin a ka sebeletsa e le tsepisa phekolo kgetho bakeng sa mafu a dikopanothutano tse kang lefu la Alzheimer le ho mefuta e meng ea 'dementia'.

3. Icariin ke Neuroprotective le e Khothalletsa Neurogenesis

Icariin thibela neurotoxicity hlohlelletsoa ke corticosterone, aluminium, peroxide hydrogen, 'me chefo e meng' me e khothalletsa neuronal pholoha ka dikai tse ngata phoofolo.

Icariin ile a fumanoa a ho thibela neurotoxicity ka ho lula intracellular k'halsiamo homeostasis ka methapo ea kutlo Rat hippocampal.

Icariin ile a boela a fumana ho thibela metsoako β-amyloid-hlohlelletsoa neurotoxicity (by eketseha ho reka (k'hok'heine le entsoeng ka amphetamine-laolwa tlaleho) liseleng cortical neuron). Fumanoa hohle boko, CARTfunctions ho thibela ho lahleheloa ke matla le ho boloka mosebetsi mitochondrial.

Mitochondria li tsejoa ho bapala karolo ea bohlokoa ho eketsa tlhahiso ea matla bakeng sa ho pholoha neuronal nakong setorouku ka.

Icariin hape khothalletsa neuronal pholoha nakong eo ho leqeba ke eketseha Sirtuin 1 (SIRT1), e potlakisang tsebetso ea lik'hemik'hale hore khothalletsa lisele khatello ea kelello ho hanyetsa.

SIRT1 activates le PGC-1alpha tseleng, e tsebahalang ho kgothaletsa mitochondrial biogenesis le metabolism matla.

Hape, SIRT1 ka fokotsa khatello ea kelello oxidative, le Ntho e ka sehloohong amehang protheine le DNA tsenyo e seleng.

Icariin di hlohleletsago neurogenesis ke activating le tape lisele tse bakoang neural ka lithuto tsa liphoofolo.

4. lowers Khatello ea Kelello le Melao e Antidepressant e

The HPA (hypothalamic-pituitary-adrenal) selekane phetha karolo ea ka go fokotsa likarabo fisioloji ho khatello ea kelello, le hyperactivity nkha lefotha ka tepelletsang le matšoenyeho maloetse.

Icariin normalizes HPA selekane mosebetsi (ka ho fokotsa CRF le ea tse ling IL-6 le TNF-alpha,) ka jpeg (sa foleng le bonolo ho imeloa kelellong) Rat dikai.

Ea tse ling IL-6 le TNF-alpha, ebe o kenya tshebetsong CRF, e leng eketsa HPA selekane mosebetsi tšoauoa ka maemo a phahameng a cortisol, e tlas'a khatello ea kelello-hormone.

Ka tsela eo icariin e ka sebetsa jwalo ka antidepressant e ka fokotseha HPA selekane hyperactivity ka thibelo ya CRF le cytokine maemo bakuli tepelletsang

5. di hlohleletsago Bone Kgolo le Repair

tse ngata tsa liphuputso li bontša hore icariin kgothaletsa kgolo ya bone bone le ho lokisa ka Stimulating lesapo (osteoblast) (lesapo eaba ba etsa) mosebetsi le inhibiting osteoclastic (thipitlo lesapo) mosebetsi.

Icariin eketsehileng noka ka tlaase le lesapo la mokokotlo lesapo segokanyipalo ka basali postmenopausal ke inhibiting felisoeng ha lesapo (lesapo heletsa) lesupa deoxypyridinoline le boloka osteocalcin, lesapo sebopeho lesupa.

Icariin ntlafatsa lesapo matsoai segokanyipalo le matla ka likhoto e motšehali le mae a bomme tlositse.

Icariin ka boela ho kgothaletsa tlhahiso le mosebetsi oa lesapo (osteoblast) liseleng.

Icariin susumelletseha ho moloko oa batho bone bone rutehileng (osteoblast) lisele tse ka eketseha lesapo morphogenetic protheine (BMP-2) tlhahiso, protheine senotlolo amehang lesapo le lefufuru sebopeho.

Icariin ile a boela a fumana ho ntlafatsa tlhahiso ea osteoblasts mathomo (by eketseha lesapo sebopeho batshwai ALP, osteocalcin, BAKOL-1 le OPG le fokotseha RANKL, protheine amehang osteoclast sebopeho).

Icariin thibela sebopeho le masapo-resorbing bohato ba osteoclasts ke eketseha dikabo OPG / RANKL liseleng masapo.

Osteoprotegerin (OPG) tsejoa ho thibela metsoako mosebetsi RANKL eo phetha karolo ea ka osteoclast sebopeho le ho timetsoa ha masapo.

Ho phaella moo, Icariin ka thibela osteoclast sebopeho ke fokotseha superoxides, mefuta oksijene arabelang hore lia hlokahala bakeng sa osteoclast ho pholoha le mosebetsi.

Icariin ka thibela metsoako lefufuru le masapo tlontlollong ka litoeba ramatiki (by inhibiting cathepsin K, e potlakisang tsebetso ea lik'hemik'hale hore roba fatše lefufuru le masapo).

6. e Khothalletsa Heart Bophelo

Icariin hlahisa liphello pelo le sireletsang lithuto tse ngata tsa liphoofolo.

Icariin ntlafala pelo mosebetsi le fokotswa lefu dinama tse nyenyane tse ka likhoto le pelo e tlhaselo hlobaetsang (myocardial infarction) ke activating le PI3K-Akt tseleng, tseo o phetha karolo ea bohlokoa ka ho pholoha seleng.

Icariin thibela pelo mesifa seleng ea lefu nakong reoxygenation latelang e hlobaetsang pelo tlhaselo ke eketseha Bc1-2 (e-ba khahlanong le tsona seleng e lefu Ntlha e) le fokotseha Bax (a lan-seleng ea lefu Ntlha e). liphello tsena ke karolo e itseng ka lebaka la ho Tshebediso ya ya PI3K / Akt tseleng, e leng eketsa Bc1-2 liseleng pelo mesifa.

Ka ho ithuta e 'ngoe, icariin thibang pelo mesifa seleng ea lefu ka ho hatella popeho metalloproteinase (MMP) mosebetsi ka likhoto le ha pelo. MMPs ke enzyme ameha pelo ntlafatsoa ha mohaho oo ka mor'a kotsi.

Icariin ntlafala pelo mosebetsi ka ho fokotsa tšenyo e oxidative ka mitochondria a lipelo tsa lefu la tsoekere Rat. Icariin ntlafatsa phallo ea mali ka ho teba ka ho atolosa lijana pelo ka tsela thibelo ea Ca2 + metjha e, e thusang ho fokotsa kotsi ya pelo leqeba le lefu dinama tse nyenyane tse.

Satalatsa tsa methapo (atherosclerosis) ke sesosa le tloaelehileng la leqeba le lefu la pelo. Icariin ka fokotsa menyetla ea thatafatsa ea methapo ka theola maemo k'holeseterole maling.

lithuto tse ngata li bontša hore icariin ka ho kgothaletsa e ncha sebopeho pelo mesifa seleng ea ka ho susumelletsa lefu seleng, eketsa arabelang oksijene mefuta molokong o mong ka, le activating e P38 MAPK le NF-kappaB litseleng ka toeba lisele tse bakoang embryonic, e leng se bontšang hore icariin ka 'na na le kopo bokgoni ba ka dinama tse nyenyane tse pelo boenjiniere.

7. di hlohleletsago sebopeho Mali Sejana

New mali sejana sebopeho ntlafatsa likotsi leqeba amanang dinama tse nyenyane tse 'me qetellong ke pholiso ke eketseha oksijene le limatlafatsi tse ngata ho sebakeng se amehileng.

Icariin ka susumelletsa kgolo ya mali sejana (by activating le Mek / ERK le PI3K / Akt / eNOS litseleng) liseleng batho mali sejana. litseleng tsena li amahanngoa le moloko, motsamao le mehaho laoleng ea lisele tsa mali sejana nakong kgolo ya mali sejana.

8. hlahisa Anti-Kankere Liphello

Icariin thibela hlahala le thehoa ka mefuta e sa tšoaneng ea kankere, ho akarelletsa le kankere ea matsoele, kankere ea mali, Burkitt lymphoma, le kankere ea sebete.

Liseleng bolaoa ke kankere ka mpeng ea batho, icariin o ile a khona ho thibela mokhatlo oa hlahala sele le tlhaselo (by inhibiting le Rac1-itšetlehileng ka VASP tseleng, tseo ho akarelletsa motility lisele).

ho ithuta e 'ngoe o ile a bontša hore Icariin o ile a khona ho thibela ikamahanya le motsamao oa lisele tsa stomachcancer (by inactivation tsa protheine kinase A (PKA), e potlakisang tsebetso ea lik'hemik'hale ho tsejoe ke ho kgothaletsa ho hlahisoeng sele le ho pholoha).

Icariin thibang batho tlhahiso ea gallbladder bolaoa ke kankere ka sele le hlohlelletsoa lefu seleng ea ka ho hatella NF-κB mosebetsi. The NF-KB tseleng phetha karolo ea bohlokoa ka ho pholoha bakeng sa kankere seleng ea ka ho eketseha-ba khahlanong le tsona seleng e lefu lintlha survivin le Bc1.

Icariin tsosa batho bakeng sa kankere sebete seleng ea lefu (by activating le Ros / JNK-itšetlehileng ka mitochondrial tseleng eo phetha karolo ea bohlokoa ka ho qapa lefu seleng e).

9. Icariin ke Anti-a hlabang le Immunoprotective

Icariin o ile a khona ho fokotsa mala ho ruruha le ntlafatsa matšoao a lefu ka litoeba le ho teneha feela mantle a syndrome, (ke thibelo ea STAT1 le STAT3 phosphorylation eo ke nang le boikarabelo bakeng sa activating le ho eketseha 1akir le Th17 T-lisele le ea tse ling lan-hlabang).

Icariin ntlafala airway ruruha ka likhoto asthmatic (by fetola ho 1akir / 2akir cytokine imbalance ka dinama tse nyenyane tse ea matšoafo). Icariin hape thibang ho Tshebediso ya ya NF-κB tseleng ka dinama tse nyenyane tse ea matšoafo, e leng ka setotsoana ho ruruha.

ho ithuta e 'ngoe o ile a bontša hore icariin fokotseha ho ruruha ea matšoafo (by inhibiting lan-hlabang batshwai TNF-α, IL-6, Cox-2 le iNOS ka ea matšoafo le ka tsela e kenngwe tshebetsong ya PI3K / Akt tseleng le thibelo ya NF-κB).

Icariin eketsa tlhahiso ea ba nyahamisa-joaloka receptor 9 (TLR9) ka macrophages toeba. TLR9 ke protheine le sebetsang ka pathogen ho amohela le Tshebediso ya a ka karabelo boitshireletso tlhaho.

Multiple sclerosis (MS) ke autoimmune lefu leo ​​ho lona T-lisele tse hlasela ba ka boko ba tsamaiso ea methapo (CNS), a etsa hore axon tshenyo le bokooa. Icariin ile a fumanoa a ho ntlafatsa matšoao a lefu ka litoeba le hlohlelletsoa MS (by hatella tlhahiso ea lisele tse T le 1akir le Th17 lisele tse).

10. Na Loantša Mokhathala

Phuputso e ile ea bontša hore icariin o ile a khona ho fokotsa mokhathala 'meleng le eketsa mamello litoeba nakong ea boima ba' mele laela teko sesa.

Ho ile ha fumanoa hore icariin eketseha tsoekere mali, haemoglobin le glycogen maemo, lintlha tse tsebahalang ho ntlafatsa lebelo, mamello le bokhoni ba ho ikoetlisa.

Icariin hape fokotseha mali lactic acid e (BLA) le mali urea naetrojene (Bun) maemo bontšang hore icariin ka 'na fokotsa le protheine thipitlo bakeng sa matla le lieha buildup ea acid e lactic, lintlha ka bobeli tsebahalang ho thibela mokhathala.

11. Sireletsa DNA le tieho ho Tsofala

Icariin sireletsa DNA tlisoang khōlō-hlohlelletsoa ka ho fokotsa tšenyo e oxidative (ka ho eketseha SIRT1 le antioxidant enzyme Cat le Prx1).

tieho Icariin botsofali ka litoeba ke eketseha SIRT6. SIRT6 ke potlakisang tsebetso ea lik'hemik'hale hore khothalletsa DNA ho lokisa le metabolism matla le thibela ho NF-KB tseleng, tseo ho akarelletsa botsofali lisele, lefu, 'me ho ruruha.

Icariin hape tieho botsofali ka libōkō ka ho khothalletsa ho imeloa kelellong ho hanyetsa, mosebetsi mesifa, 'me mokhatlo oa,' me ho thibela protheine haha ​​toxicity.

12. Na Thusa maqoqomete a makhopho

Phuputso e ile ea bontša hore Icariin ile a khona ho thibela metsoako Propionibacterium acnes biofilm sebopeho e sa fella ka ho bolaea lisele baktheria. Propionibacterium acnes ke baktheria e amana le boemo ba letlalo la maqoqomete, e leng se bontšang hore icariin e ka sebelisoa e le mokhoa oa tlhaho-ba khahlanong le maqoqomete lithethefatsi.

13. Na Thusa pele ho nako mora ho ntsha peo

Ka habeli-ba foufetseng, ea lotho teko taolo, PDE5 inhibitors ka lelefatsa nako eo ho nka ho ejaculate.

14. Na Fight Jetlag

PDE5 inhibitors ntlafatsa likarabo circadian leseling le fokotseha ka nako eo ho hlokahala hore botjha entrainment ka litoeba.

Sena se thusa ha u fofa ka nģ'a bochabela. Nka hore u fofa bochabela 3 nako libaka tloha California ho ea New York.

Nka hore u fofa bochabela 3 nako libaka tloha California ho ea New York. Haeba u ka tloaelo robala ka 11 PM California nako, ka nako eo o tla il'o robala ho 2 AM New York nako.

Haeba u batla ho ea robala ka eena pejana, o lokela ho tsoha pejana ho moo, le 'pele' potoloho hao e le hore u robala pejana, 'me o tsoha pejana.

Icariin le PDE5 inhibitors u thusa ho ntshetsa pele morethetho oa hao. Sheba hlahlobeloa ea ka le ea ka mongoli oa sehlooho sena se.


Post nako: Sep-01-2019
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