CAS No .: 5508-58 -7
Igama Lesi'Latin: Andrographis paniculata (Burm.f) Ness
Ingxenye esetshenziswa: lonke imbiza
Ukubukeka: ukukhanya yellow ukuba powder emhlophe
Formula Yamamolekhula: C20H 30O 5
Isisindo Yamamolekhula: 350,455
Indlela Test: HPLC
Ukucaciswa:
Andrographolide50%
Andrographolide98%
Andrographolide99%
Andrographolide kuyinto diterpenoid labdane okungukuthi main ingxenye bioactive A. paniculata, kahle neyaziwayo isitshalo okwelapha e-Asia. It siba ezahlukene izenzo zokwelapha, kuhlanganise immunosuppressant, antithrombotic, eqeda ukuvuvukala, antineoplastic, elwa namagciwane, elwa namagciwane, antidiabetic, ukucindezeleka antioxidative, antipyretic, antioedematogenic, futhi antinociceptive ukwelashwa activities.1Andrographolide kuvimbela isici yenuzi kappa B (NF-κB) iyawabopha ukuze abagqugquzeli DNA target izakhi zofuzo (IC50 = ~ 15 μM), ngokwakha adduct covalent nge cysteine encishisiwe (62) we-NF-κB p50 subunit, futhi ungakwazi futhi ntombazane inkulumo subfamily CYP1A omkhaya cytochrome P450 enzyme. 2,3 Ngezinye 5 μg g isisindo / umzimba kungenza yokuvimbela ukusebenza NF-κB kumaseli uyavuselelwa endothelial, ukunciphisa ukubonakaliswa iseli adhesion-molecule e-selectin, abrogating le cytokine- futhi endotoxin olubangelwa kokuziphatha peritoneal ka neutrophil nama attenuating ukushaqeka ukonakala, nokuvimbela iguliswa wamaphaphu ukuvuvukala endaweni imodeli igundane of asthma.3
Umkhiqizo nokupakisha: 25kg / isigubhu
Isikhathi Ukuhlola ngokuqinisekisa: iminyaka engu-2